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Tracazolate hydrochloride
CAS No. 1135210-68-2
Tracazolate hydrochloride ( Tracazolate (hydrochloride) )
Catalog No. M27728 CAS No. 1135210-68-2
Tracazolate hydrochloride is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 32 | Get Quote |
|
| 5MG | 53 | Get Quote |
|
| 10MG | 86 | Get Quote |
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| 25MG | 177 | Get Quote |
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| 50MG | 295 | Get Quote |
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| 100MG | 444 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameTracazolate hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionTracazolate hydrochloride is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.
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DescriptionTracazolate hydrochloride is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity. Tracazolate hydrochloride potentiates α1β1γ2s and α1β3γ2 with EC50s of 13.2 μM and 1.5 μM.(In Vitro):Tracazolate hydrochloride (10 μM) enhanced the sensitivity of α1β2δ-containing GABAA receptors and increased the maximum current amplitude in oocytes . Tracazolate hydrochloride inhibited α1β1ε, α1β3ε, α1β3, and α6β3γ with EC50s of 4.0 μM, 1.2 μM, 2.7 μM, and 1.1 μM. Tracazolate hydrochloride interacted with γ-aminobutyric acid GABAA receptors, adenosine receptors, and phosphodiesterases .
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SynonymsTracazolate (hydrochloride)
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PathwayOthers
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TargetOther Targets
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number1135210-68-2
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Formula Weight340.9
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Molecular FormulaC16H25ClN4O2
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Purity>98% (HPLC)
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Solubility——
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SMILESCl.CCCCNc1c(C(=O)OCC)c(C)nc2n(CC)ncc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.King HL Jr, Dyar RE, Wilken DR. Ketopantoyl lactone and ketopantoic acid reductases. Characterization of the reactions and purification of two forms of ketopantoyl lactone reductase. J Biol Chem. 1974 Aug 10;249(15):4689-95.
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